A novel 4-aminoquinoline chemotype with multistage antimalarial activity and lack of cross-resistance with PfCRT and PfMDR1 mutants

Ferreira, L. T., Cassiano, G. C., Alvarez, L. C. S., Okombo, J., Calit, J., Fontinha, D., Gil-Iturbe, E., Coyle, R., Andrade, C. H., Sunnerhagen, P., Bargieri, D. Y., Prudêncio, M., Quick, M., Cravo, P. V., Lee, M. C. S., Fidock, D. A., & Costa, F. T. M. (2024). A novel 4-aminoquinoline chemotype with multistage antimalarial activity and lack of cross-resistance with PfCRT and PfMDR1 mutants. PLOS Pathogens, 20(10), e1012627. https://doi.org/10.1371/journal.ppat.1012627
Authors:
Letícia Tiburcio Ferreira
Gustavo Capatti Cassiano
Luis Carlos Salazar Alvarez
John Okombo
Juliana Calit
Diana Fontinha
Eva Gil-Iturbe
Rachael Coyle
Carolina Horta Andrade
Per Sunnerhagen
Daniel Youssef Bargieri
Miguel Prudêncio
Matthias Quick
Pedro V Cravo
Marcus C S Lee
David A Fidock
Fabio Trindade Maranhão Costa
Affiliated Authors:
Letícia Tiburcio Ferreira
John Okombo
Eva Gil-Iturbe
Matthias Quick
David A Fidock
Publication Type:
Article
Unique ID:
10.1371/journal.ppat.1012627
PMID:
Journal:
Publication Date:
Data Source:
PubMed

Record Created: