European Journal of Medicinal Chemistry
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Awalt, J. K., Su, W., Nguyen, W., Loi, K., Jarman, K. E., Penington, J. S., Ramesh, S., Fairhurst, K. J., Yeo, T., Park, H., Uhlemann, A.-C., Chandra Maity, B., De, N., Mukherjee, P., Chakraborty, A., Churchyard, A., Famodimu, M. T., Delves, M. J., Baum, J., … Sleebs, B. E. (2024). Exploration and characterization of the antimalarial activity of cyclopropyl carboxamides that target the mitochondrial protein, cytochrome b. European Journal of Medicinal Chemistry, 280, 116921. https://doi.org/10.1016/j.ejmech.2024.116921
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Calic, P. P. S., Ashton, T. D., Mansouri, M., Loi, K., Jarman, K. E., Qiu, D., Lehane, A. M., Roy, S., Rao, G. P., Maity, B., Wittlin, S., Crespo, B., Gamo, F.-J., Deni, I., Fidock, D. A., Chowdury, M., de Koning-Ward, T. F., Cowman, A. F., Jackson, P. F., … Sleebs, B. E. (2024). Optimization of pyrazolopyridine 4-carboxamides with potent antimalarial activity for which resistance is associated with the P. falciparum transporter ABCI3. European Journal of Medicinal Chemistry, 276, 116677. https://doi.org/10.1016/j.ejmech.2024.116677
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Nguyen, W., Boulet, C., Dans, M. G., Loi, K., Jarman, K. E., Watson, G. M., Tham, W.-H., Fairhurst, K. J., Yeo, T., Fidock, D. A., Wittlin, S., Chowdury, M., de Koning-Ward, T. F., Chen, G., Yan, D., Charman, S. A., Baud, D., Brand, S., Jackson, P. F., … Sleebs, B. E. (2024). Activity refinement of aryl amino acetamides that target the P. falciparum STAR-related lipid transfer 1 protein. European Journal of Medicinal Chemistry, 270, 116354. https://doi.org/10.1016/j.ejmech.2024.116354
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Al Noman, M. A., Cuellar, R. A. D., Kyzer, J. L., Chung, S. S. W., Cheryala, N., Holth, T. A. D., Maitra, S., Naqvi, T., Wong, H. L., Schönbrunn, E., Hawkinson, J. E., Wolgemuth, D. J., & Georg, G. I. (2023). Strategies for developing retinoic acid receptor alpha-selective antagonists as novel agents for male contraception. European Journal of Medicinal Chemistry, 261, 115821. https://doi.org/10.1016/j.ejmech.2023.115821
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Mehta, V., Dwivedi, A. R., Ludhiadch, A., Rana, V., Goel, K. K., Uniyal, P., Joshi, G., Kumar, A., & Kumar, B. (2024). A decade of USFDA-approved small molecules as anti-inflammatory agents: Recent trends and Commentaries on the “industrial” perspective. European Journal of Medicinal Chemistry, 263, 115942. https://doi.org/10.1016/j.ejmech.2023.115942
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Lin, W., Gandhi, S., Bhattarai, P., Kasa, K., Kizil, C., & Zhang, Y. (2023). Combining high throughput array synthesis and growth algorithm to discover TNF-α binders with new structures and properties. European Journal of Medicinal Chemistry, 248, 115078. https://doi.org/10.1016/j.ejmech.2022.115078
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Columbia Affiliation