Calic, P. P. S., Ashton, T. D., Mansouri, M., Loi, K., Jarman, K. E., Qiu, D., Lehane, A. M., Roy, S., Rao, G. P., Maity, B., Wittlin, S., Crespo, B., Gamo, F.-J., Deni, I., Fidock, D. A., Chowdury, M., de Koning-Ward, T. F., Cowman, A. F., Jackson, P. F., … Sleebs, B. E. (2024). Optimization of pyrazolopyridine 4-carboxamides with potent antimalarial activity for which resistance is associated with the P. falciparum transporter ABCI3. European Journal of Medicinal Chemistry, 276, 116677. https://doi.org/10.1016/j.ejmech.2024.116677
Subjects:
Malaria
(OpenAlex Topic)
Mechanisms of Multidrug Resistance in Cancer
(OpenAlex Topic)
Efficacy and Safety of Antiretroviral Therapy for HIV
(OpenAlex Topic)
Antimalarials
(MeSH)
Plasmodium falciparum
(MeSH)
Pyrazoles
(MeSH)
Pyridines
(MeSH)
Publication Type:
Article
Unique ID:
10.1016/j.ejmech.2024.116677
PMID:
Publication Date:
Data Source:
PubMed