Optimization of pyrazolopyridine 4-carboxamides with potent antimalarial activity for which resistance is associated with the P. falciparum transporter ABCI3

Calic, P. P. S., Ashton, T. D., Mansouri, M., Loi, K., Jarman, K. E., Qiu, D., Lehane, A. M., Roy, S., Rao, G. P., Maity, B., Wittlin, S., Crespo, B., Gamo, F.-J., Deni, I., Fidock, D. A., Chowdury, M., de Koning-Ward, T. F., Cowman, A. F., Jackson, P. F., … Sleebs, B. E. (2024). Optimization of pyrazolopyridine 4-carboxamides with potent antimalarial activity for which resistance is associated with the P. falciparum transporter ABCI3. European Journal of Medicinal Chemistry, 276, 116677. https://doi.org/10.1016/j.ejmech.2024.116677
Authors:
Petar P S Calic
Trent D Ashton
Mahta Mansouri
Katie Loi
Kate E Jarman
Deyun Qiu
Adele M Lehane
Sayantan Roy
Gunturu P Rao
Bikash Maity
Sergio Wittlin
Benigno Crespo
Franciso-Javier Gamo
Ioanna Deni
David A Fidock
Mrittika Chowdury
Tania F de Koning-Ward
Alan F Cowman
Paul F Jackson
Delphine Baud
Stephen Brand
Benoît Laleu
Brad E Sleebs
Affiliated Authors:
Ioanna Deni
David A Fidock
Author Keywords:
abci3 transporter
antimalarial
malaria
plasmodium
pyrazolopyridine
Publication Type:
Article
Unique ID:
10.1016/j.ejmech.2024.116677
PMID:
Publication Date:
Data Source:
PubMed

Record Created: