Optimization of 2,3-Dihydroquinazolinone-3-carboxamides as Antimalarials Targeting PfATP4

Ashton, T. D., Dans, M. G., Favuzza, P., Ngo, A., Lehane, A. M., Zhang, X., Qiu, D., Chandra Maity, B., De, N., Schindler, K. A., Yeo, T., Park, H., Uhlemann, A.-C., Churchyard, A., Baum, J., Fidock, D. A., Jarman, K. E., Lowes, K. N., Baud, D., … Sleebs, B. E. (2023). Optimization of 2,3-Dihydroquinazolinone-3-carboxamides as Antimalarials Targeting PfATP4. Journal of Medicinal Chemistry, 66(5), 3540–3565. https://doi.org/10.1021/acs.jmedchem.2c02092
Authors:
Trent D Ashton
Madeline G Dans
Paola Favuzza
Anna Ngo
Adele M Lehane
Xinxin Zhang
Deyun Qiu
Bikash Chandra Maity
Nirupam De
Kyra A Schindler
Tomas Yeo
Heekuk Park
Anne-Catrin Uhlemann
Alisje Churchyard
Jake Baum
David A Fidock
Kate E Jarman
Kym N Lowes
Delphine Baud
Stephen Brand
Paul F Jackson
Alan F Cowman
Brad E Sleebs
Affiliated Authors:
Kyra A Schindler
Tomas Yeo
Heekuk Park
Anne-Catrin Uhlemann
David A Fidock
Publication Type:
Article
Unique ID:
10.1021/acs.jmedchem.2c02092
PMID:
Publication Date:
Data Source:
PubMed

Record Created: