TKK130 is a 3-Hydroxy-Propanamidine (HPA) with Potent Antimalarial In Vivo Activity and a High Barrier to Resistance

Knaab, T. C., Moritz, A., Pessanha de Carvalho, L., Klein, S., Lungerich, B., Lohse, K., Kruse, L., Mombo-Ngoma, G., Orta, L., Thibaud, J. L., de Villiers, K. A., Fidock, D. A., Burckhardt, B. B., Held, J., Wittlin, S., & Kurz, T. (2024). TKK130 is a 3-Hydroxy-Propanamidine (HPA) with Potent Antimalarial In Vivo Activity and a High Barrier to Resistance. Journal of Medicinal Chemistry. https://doi.org/10.1021/acs.jmedchem.4c01465
Authors:
Tanja C Knaab
Alena Moritz
Lais Pessanha de Carvalho
Saskia Klein
Beate Lungerich
Katharina Lohse
Linn Kruse
Ghyslain Mombo-Ngoma
Lily Orta
Jessica L Thibaud
Katherine A de Villiers
David A Fidock
Bjoern B Burckhardt
Jana Held
Sergio Wittlin
Thomas Kurz
Affiliated Authors:
Lais Pessanha de Carvalho
Lily Orta
David A Fidock
Publication Type:
Article
Unique ID:
10.1021/acs.jmedchem.4c01465
PMID:
Publication Date:
Data Source:
PubMed

Record Created: