A Novel Mitragynine Analog with Low-Efficacy Mu Opioid Receptor Agonism Displays Antinociception with Attenuated Adverse Effects

Chakraborty, S., DiBerto, J. F., Faouzi, A., Bernhard, S. M., Gutridge, A. M., Ramsey, S., Zhou, Y., Provasi, D., Nuthikattu, N., Jilakara, R., Nelson, M. N. F., Asher, W. B., Eans, S. O., Wilson, L. L., Chintala, S. M., Filizola, M., van Rijn, R. M., Margolis, E. B., Roth, B. L., … Majumdar, S. (2021). A Novel Mitragynine Analog with Low-Efficacy Mu Opioid Receptor Agonism Displays Antinociception with Attenuated Adverse Effects. Journal of Medicinal Chemistry, 64(18), 13873–13892. https://doi.org/10.1021/acs.jmedchem.1c01273
Authors:
Soumen Chakraborty
Jeffrey F DiBerto
Abdelfattah Faouzi
Sarah M Bernhard
Anna M Gutridge
Steven Ramsey
Yuchen Zhou
Davide Provasi
Nitin Nuthikattu
Rahul Jilakara
Melissa N F Nelson
Wesley B Asher
Shainnel O Eans
Lisa L Wilson
Satyanarayana M Chintala
Marta Filizola
Richard M van Rijn
Elyssa B Margolis
Bryan L Roth
Jay P McLaughlin
Tao Che
Dalibor Sames
Jonathan A Javitch
Susruta Majumdar
Affiliated Authors:
Melissa N F Nelson
Wesley B Asher
Jonathan A Javitch
Publication Type:
Article
Unique ID:
10.1021/acs.jmedchem.1c01273
PMID:
Publication Date:
Data Source:
PubMed

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