Site selective C–H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy

Bhowmik, S., Galeta, J., Havel, V., Nelson, M., Faouzi, A., Bechand, B., Ansonoff, M., Fiala, T., Hunkele, A., Kruegel, A. C., Pintar, John. E., Majumdar, S., Javitch, J. A., & Sames, D. (2021). Site selective C–H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy. Nature Communications, 12(1). https://doi.org/10.1038/s41467-021-23736-2
Authors:
Srijita Bhowmik
Juraj Galeta
Václav Havel
Melissa Nelson
Abdelfattah Faouzi
Benjamin Bechand
Mike Ansonoff
Tomas Fiala
Amanda Hunkele
Andrew C. Kruegel
John. E. Pintar
Susruta Majumdar
Jonathan A. Javitch
Dalibor Sames
Affiliated Authors:
Juraj Galeta
Melissa Nelson
Jonathan A. Javitch
Dalibor Sames
Publication Type:
Article
Unique ID:
10.1038/s41467-021-23736-2
PMID:
Publication Date:
Data Source:
Scopus

Record Created: