Activity refinement of aryl amino acetamides that target the P. falciparum STAR-related lipid transfer 1 protein

Nguyen, W., Boulet, C., Dans, M. G., Loi, K., Jarman, K. E., Watson, G. M., Tham, W.-H., Fairhurst, K. J., Yeo, T., Fidock, D. A., Wittlin, S., Chowdury, M., de Koning-Ward, T. F., Chen, G., Yan, D., Charman, S. A., Baud, D., Brand, S., Jackson, P. F., … Sleebs, B. E. (2024). Activity refinement of aryl amino acetamides that target the P. falciparum STAR-related lipid transfer 1 protein. European Journal of Medicinal Chemistry, 270, 116354. https://doi.org/10.1016/j.ejmech.2024.116354
Authors:
William Nguyen
Coralie Boulet
Madeline G Dans
Katie Loi
Kate E Jarman
Gabrielle M Watson
Wai-Hong Tham
Kate J Fairhurst
Tomas Yeo
David A Fidock
Sergio Wittlin
Mrittika Chowdury
Tania F de Koning-Ward
Gong Chen
Dandan Yan
Susan A Charman
Delphine Baud
Stephen Brand
Paul F Jackson
Alan F Cowman
Paul R Gilson
Brad E Sleebs
Affiliated Authors:
Kate J Fairhurst
Tomas Yeo
David A Fidock
Subjects:
Author Keywords:
malaria
plasmodium
antimalarial
star lipid transfer
aryl amino acetamide
Publication Type:
Article
Unique ID:
10.1016/j.ejmech.2024.116354
PMID:
Publication Date:
Data Source:
PubMed

Record Created: