Bioorganic and Medicinal Chemistry Letters

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Zuccarello, E., Zhang, H., Acquarone, E., Pham, D., Staniszewski, A., Deng, S.-X., Landry, D. W., Arancio, O., & Fiorito, J. (2023). Optimizing metabolic stability of phosphodiesterase 5 inhibitors: Discovery of a potent N-(pyridin-3-ylmethyl)quinoline derivative targeting synaptic plasticity. Bioorganic & Medicinal Chemistry Letters, 92, 129409. https://doi.org/10.1016/j.bmcl.2023.129409
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Dileep Kumar, J. S., Molotkov, A., Carberry, P., Chaly, T., Neelamegam, R., & Mintz, A. (2022). Radiosynthesis and evaluation of [11C]AG-488, a dual anti-angiogenetic and anti-tubulin PET ligand. Bioorganic & Medicinal Chemistry Letters, 74, 128941. https://doi.org/10.1016/j.bmcl.2022.128941
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