Positive and negative allosteric modulation of GluK2 kainate receptors by BPAM344 and antiepileptic perampanel

Gangwar, S. P., Yen, L. Y., Yelshanskaya, M. V., & Sobolevsky, A. I. (2023). Positive and negative allosteric modulation of GluK2 kainate receptors by BPAM344 and antiepileptic perampanel. Cell Reports, 42(2), 112124. https://doi.org/10.1016/j.celrep.2023.112124
Authors:
S.P. Gangwar
Laura Y. Kim
M.V. Yelshanskaya
Alexander I. Sobolevsky
Affiliated Authors:
S.P. Gangwar
Laura Y. Kim
M.V. Yelshanskaya
Alexander I. Sobolevsky
Columbia Affiliation:
Subjects:
Anticonvulsants (MeSH)
Receptors, Kainic Acid (MeSH)
Molecular Mechanisms of Synaptic Plasticity and Neurological Disorders (OpenAlex Topic)
Lipid Rafts and Membrane Dynamics (OpenAlex Topic)
Molecular Mechanisms of Ion Channels Regulation (OpenAlex Topic)
Author Keywords:
bpam344
competitive antagonist
cp: molecular biology
cp: neuroscience
cryo-em
dnqx
gluk2
iglur
kainate receptor
negative allosteric modulator
perampanel
positive allosteric modulator
elink
Publication Type:
Article
Unique ID:
10.1016/j.celrep.2023.112124
PMID:
36857176
DOI:
10.1016/j.celrep.2023.112124
Journal:
Cell Reports
Publication Date:
Data Source:
OpenAlex
Source Link:
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Record Created: