Discovery of Indole-Based PDE5 Inhibitors: Synthesis and Pharmacological Evaluation

Park, S.-Y., Pham, D., Shukla, P., Edward, J., John, R., Li, A., Hadjiargyrou, M., Mori, M., Zuccarello, E., Arancio, O., & Fiorito, J. (2025). Discovery of Indole-Based PDE5 Inhibitors: Synthesis and Pharmacological Evaluation. ACS Medicinal Chemistry Letters, 16(6), 1058–1065. https://doi.org/10.1021/acsmedchemlett.5c00108
Authors:
Shin-Young Park
Dang Pham
Param Shukla
Justin Edward
Reshmi John
Addison Li
Michael Hadjiargyrou
Mattia Mori
Elisa Zuccarello
Ottavio Arancio
Jole Fiorito
Affiliated Authors:
Elisa Zuccarello
Ottavio Arancio
Jole Fiorito
Author Keywords:
alzheimer’s disease
indole-containing molecules
pde5
pde5 inhibitors
Publication Type:
Article
Unique ID:
10.1021/acsmedchemlett.5c00108
PMID:
Publication Date:
Data Source:
PubMed

Record Created: